Question

On an inhibition curve, the IC50 for an antagonist is seen to be directly above the number 8 on the x-axis, which is labeled -Log(drug). What concentration of drug is the IC50? in M in nM 2. Corrected_text: For the drug in Q1, above, what PERCENT of the receptors is occupied by the antagonist when the concentration on the inhibition curve is directly above the number 9? 3. Corrected_text: For the drug in Q1, above, what FRACTION of the receptors is occupied by the antagonist when the concentration on the inhibition curve is directly above the number? 4. Corrected_text: For the drug in Q1, above, if the radioligand concentration is 1 nM and the Kd of the radioligand is 0.1 nM, what is the Kd value of the drug? Specify units. Kd= 5. Corrected_text: For the antagonist drug in Q1, if the rate constant of dissociation is 0.02 per second, what is the calculated value for the rate constant of association, assuming simple reaction kinetics? Specify the units. k1=

          On an inhibition curve, the IC50 for an antagonist is seen to be directly above the number 8 on the x-axis, which is labeled -Log(drug). What concentration of drug is the IC50?
in M
in nM

2. Corrected_text: For the drug in Q1, above, what PERCENT of the receptors is occupied by the antagonist when the concentration on the inhibition curve is directly above the number 9?

3. Corrected_text: For the drug in Q1, above, what FRACTION of the receptors is occupied by the antagonist when the concentration on the inhibition curve is directly above the number?

4. Corrected_text: For the drug in Q1, above, if the radioligand concentration is 1 nM and the Kd of the radioligand is 0.1 nM, what is the Kd value of the drug? Specify units.
Kd=

5. Corrected_text: For the antagonist drug in Q1, if the rate constant of dissociation is 0.02 per second, what is the calculated value for the rate constant of association, assuming simple reaction kinetics? Specify the units.
k1=

1on an inhibition curvethe ic50 for an antagonist is seen to be directly above the number 8 on the x axiswhich is labeled logdrug what concentration of drug is the ic50 in m in nm 2 for the 11697

Added by Blake S.

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